14-Ethoxymetopon

drugbox
IUPAC_name = 3-hydroxy-14-ethoxy-5-methyl-7,8-dihydro-4,5α-epoxy-17-methylmorphinan-6-one

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CAS_number = 131575-04-7
synonyms = 14-Ethoxymetopon
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PubChem = 5487378
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C = 20 | H = 25 | N = 1 | O = 4
molecular_weight = 343.42 g/mol
smiles = CCOC12CCC(=O) [C@@] 3(C14CCN( [C@@H] 2CC5=C4C(=C(C=C5)O)O3)C)C
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14-Ethoxymetopon is an opiate analogue that is an derivative of metopon which has been substituted with an ethoxy group at the 14-position. It is a highly potent analgesic drug several hundred times stronger than morphine. [Fürst Z, Búzás B, Friedmann T, Schmidhammer H, Borsodi A. Highly potent novel opioid receptor agonist in the 14-alkoxymetopon series. "European Journal of Pharmacology". 1993 May 19;236(2):209-15. PMID 8391457]

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