Burimamide

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IUPACName= 1- [4-(1H-Imidazol-5-yl)butyl] -3-methylthiourea
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CASNo=34970-69-9
PubChem=3032915
SMILES=CNC(=S)NCCCCC1=CN=CN1
Section2= Chembox Properties
Formula=C₉H₁₆N₄S
MolarMass=212.316
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Burimamide is an antagonist at the H₂ and H₃ histamine receptors. It is largely inactive as an H₂ antagonist at physiological pH, [Clayden, J. Greeves, N. Warren, S. Wothers, P. (2001). "Organic Chemistry". Oxford. ISBN 0-19-850346-6] but its H₃ affinity is 100x higher. It is a thiourea derivative.

References