CP 55,244

Drugbox
IUPAC_name = (2S,4S,4aS,6R,8aR)-6-(hydroxymethyl)-4- [2-hydroxy-4-(2-methyloctan-2-yl)phenyl] -1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-ol

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width= 240
CAS_number= 79678-32-3
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PubChem= 133254
DrugBank=
C=26 | H=42 | O=3
molecular_weight = 402.608 g/mol
smiles = C13CC(CO)CCC3CC(O)CC1c2ccc(C(C)(C)CCCCCC)cc2O
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CP 55,244 is a drug which is a cannabinoid receptor agonist. It has analgesic effects and is used in scientific research. It is a potent CB₁ full agonist with a Ki of 0.21nM, making it more potent than the commonly used full agonist HU-210. [Griffin G, Wray EJ, Martin BR, Abood ME. Cannabinoid agonists and antagonists discriminated by receptor binding in rat cerebellum. "British Journal of Pharmacology". 1999 Oct;128(3):684-8. PMID 10516649]

References