(4aR,9aS)-N-ethyl-4,4a,9,9a-tetrahydro-1H-fluoren-4a-amine

(4aR,9aS)-N-ethyl-4,4a,9,9a-tetrahydro-1H-fluoren-4a-amine

Drugbox
IUPAC_name = (4a"R",9a"S")-"N"-Ethyl-4,4a,9,9a-tetrahydro-1"H"-fluoren-4a-amine



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C=15 | H=19 | N=1
molecular_weight = 213.3181 g/mol
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NEFA is a moderate affinity NMDA antagonist (IC50 = 0.51 μM). It is a structural analog of phencyclidine. [cite journal|author=Dilmore JG, Johnson JW |title=Open channel block and alteration of N-methyl-D-aspartic acid receptor gating by an analog of phencyclidine |journal=Biophysical Journal |year=1998 |volume=75 |issue=4 |pages=1801–16]

References


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  • NEFA (drug) — Systematic (IUPAC) name (4aR,9aS) N Ethyl 4,4a,9,9a tetrahydro 1H fluoren 4a amine Clinical data Pregnancy cat …   Wikipedia

  • NEFA — is an abbreviation that has several meanings: (4aR,9aS) N ethyl 4,4a,9,9a tetrahydro 1H fluoren 4a amine The Nine Eleven Finding Answers Foundation Non essential fatty acid North East Folklore Archive North East Forest Alliance New England… …   Wikipedia

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