Cinolazepam

Not to be confused with clonazepam or camazepam.

Cinolazepam

Systematic (IUPAC) name
(RS)-3-[9-chloro- 6-(2-fluorophenyl)- 4-hydroxy- 3-oxo- 2,5-diazabicyclo [5.4.0]undeca- 5,8,10,12- tetraen- 2-yl] propanenitrile
Clinical data
AHFS/Drugs.com	International Drug Names
Pregnancy cat.	?
Legal status	IV(US)
Routes	Oral
Pharmacokinetic data
Bioavailability	90-100%
Metabolism	Hepatic
Half-life	9 h[1]
Excretion	Renal
Identifiers
CAS number	75696-02-5
ATC code	N05CD13
PubChem	CID 3033621
DrugBank	DB01594
ChemSpider	2298251 Y
UNII	68P0556B0U Y
KEGG	D07328 Y
ChEBI	CHEBI:59514 Y
Chemical data
Formula	C18H13ClFN3O2
Mol. mass	357.8
SMILES	eMolecules & PubChem
InChI InChI=1S/C18H13ClFN3O2/c19-11-6-7-15-13(10-11)16(12-4-1-2-5-14(12)20)22-17(24)18(25)23(15)9-3-8-21/h1-2,4-7,10,17,24H,3,9H2 Y Key:XAXMYHMKTCNRRZ-UHFFFAOYSA-N Y
Y(what is this?)  (verify)

Cinolazepam (marketed under the brand name Gerodorm)^[2] is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. Due to its strong sedative properties, it is primarily used as an hypnotic.

Cinolazepam is not approved for sale in the United States or Canada.

See also

• Benzodiazepine

References

1. ^ Saletu, B.; G. Kindshofer, P. Anderer, J. Grunberger (1987). "Short-term sleep laboratory studies with cinolazepam in situational insomnia induced by traffic noise.". International Journal of Clinical Pharmacology Research 7 (5): 407–18. PMID 2889679. 
2. ^ Lannacher Romania (1999). "Gerodorm" (in Romanian). Produse Gerot inregistrate in Romania. Archived from the original on 11 October 2006. http://web.archive.org/web/20061011022835/http://www.lannacher.ro/gerodorm.html. Retrieved 17 August 2006. 

External links

• Inchem.org - Cinolazepam

This sedative-related article is a stub. You can help Wikipedia by expanding it.v · Categories: Benzodiazepines Hypnotics Organochlorides Nitriles Organofluorides Lactams Alcohols Sedative stubs Wikimedia Foundation. 2010. Игры ⚽ Нужен реферат? Haplogroup C (mtDNA) Haplogroup D (mtDNA) Look at other dictionaries: Benzodiazepine — Benzodiazepines …   Wikipedia Flunitrazepam — Systematic (IUPAC) name 6 (2 …   Wikipedia Sodium thiopental — Systematic (IUPAC) name …   Wikipedia Temazepam — Systematic (IUPAC) name 7 Chloro 1,3 dihydro 3 hydroxy 1 methyl 5 phenyl 1,4 benzod …   Wikipedia Propofol — Systematic (IUPAC) name 2,6 diisopropylphenol …   Wikipedia Triazolam — Systematic (IUPAC) name 8 chloro 6 (2 chlorophenyl) 1 methyl 4H [1,2,4]triazolo[4,3 a][1,4]benzodiazepine Clinical data Tra …   Wikipedia Midazolam — Systematic (IUPAC) name 8 chloro 6 (2 fluorophenyl) 1 methyl 4H imidazo[1,5 …   Wikipedia Clonazepam — Not to be confused with camazepam, chlorpromazine, cinolazepam, or clobazam. Clonazepam …   Wikipedia Nitrazepam — Systematic (IUPAC) name …   Wikipedia Flurazepam — Systematic (IUPAC) name 7 chloro 1 [2 (diethylamino)ethyl] 5 (2 fluorophenyl) …   Wikipedia 18+ © Academic, 2000-2024 Contact us: Technical Support, Advertising Dictionaries export, created on PHP, Joomla, Drupal, WordPress, MODx. Mark and share Search through all dictionaries Translate… Search Internet Share the article and excerpts Direct link … Do a right-click on the link above and select “Copy Link”